Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with Target = 'Cannabinoid Receptor 2' and Monomerid = 50239215
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP55940 from human cloned CB2 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP 55940 from human CB2 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataKi:  34nMAssay Description:Displacement of [3H]CP-55940 from human cloned CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human cloned CB2 receptor by [35S]GTP-gamma-S binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50239215(4-methyl-3-(morpholinosulfonyl)-N-(2,2,4,4-tetrame...)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human cloned CB2 receptor assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed