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Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome Proliferator-Activated Receptor gamma' and Monomerid = 50241439
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Graduate School Of The Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50241439(2,2'-(4,4'-(propane-2,2-diyl)bis(4,1-phenylene))bi...)
Affinity DataIC50:  1.00E+5nMAssay Description:Antagonist activity at human PPARgamma receptor expressed in Saccharomyces cerevisiae AH109 co-transfected with mouse CBP assessed as inhibition of r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed