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Found 3 Enz. Inhib. hit(s) with Target = 'Apoptosis Regulator Bcl-2' and Monomerid = 50247980
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50247980(1-(2-((R)-3-(hydroxymethyl)-1,2,3,4-tetrahydroisoq...)
Affinity DataIC50:  390nMAssay Description:Inhibition of GST fused Bcl-2 (unknown origin) binding to biotinylated 16 mer BH3 peptide by HTRF-LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50247980(1-(2-((R)-3-(hydroxymethyl)-1,2,3,4-tetrahydroisoq...)
Affinity DataIC50:  390nMAssay Description:Inhibition of GST fused Bcl-2 (unknown origin) binding to biotinylated 16 mer BH3 peptide by HTRF-LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
Ucb Pharma

Curated by ChEMBL
LigandPNGBDBM50247980(1-(2-((R)-3-(hydroxymethyl)-1,2,3,4-tetrahydroisoq...)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of GST fused Bcl-2 (unknown origin) binding to biotinylated 16 mer BH3 peptide by HTRF-LANCE assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed