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Found 2 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 5' and Monomerid = 50248439
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50248439((+/-)-4,4-difluoro-N-((1S)-3-(4-(3-isopropyl-5-met...)
Affinity DataIC50:  0.840nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50248439((+/-)-4,4-difluoro-N-((1S)-3-(4-(3-isopropyl-5-met...)
Affinity DataIC50:  62nMAssay Description:Antagonist activity at human recombinant CCR5 expressed in human HeLa-P4 cells assessed as inhibition of human HeLa-P4 cells binding to HIV1 gp160 ex...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed