Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50251773
TargetProgesterone receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251773(4,4-Spirohexyl-2-(4-chlorophenyl)isoquinoline-1,3(...)
Affinity DataIC50:  1.10E+3nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251773(4,4-Spirohexyl-2-(4-chlorophenyl)isoquinoline-1,3(...)
Affinity DataIC50:  1.50E+3nMAssay Description:Antagonist activity at human progesterone receptor expressed in CHO cells assessed as inhibition of progesterone-induced luciferase activity by repor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed