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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50251799
TargetProgesterone receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251799(4-(4,4-Diallyl-3,4-dihydro-1,3-dioxoisoquinolin-2(...)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells assessed as inhibition of progesterone-induced alkaline phosphatase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50251799(4-(4,4-Diallyl-3,4-dihydro-1,3-dioxoisoquinolin-2(...)
Affinity DataIC50:  150nMAssay Description:Antagonist activity at human progesterone receptor expressed in CHO cells assessed as inhibition of progesterone-induced luciferase activity by repor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed