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Found 2 Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 3' and Monomerid = 50251894
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of [3H]D-Asp uptake at human EAAT3 in HEK293 cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExcitatory amino acid transporter 3(Homo sapiens (Human))
Universite Blaise Pascal

Curated by ChEMBL
LigandPNGBDBM50251894((2S,4R)-4-(2,2-Diphenylethylamino-3-oxopropyl)glut...)
Affinity DataIC50:  1.00E+6nMAssay Description:Inhibition of glutamate-induced depolarization in human human EAAT3 expressed in HEK293 cells by FMP assayChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed