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Found 5 Enz. Inhib. hit(s) with Target = 'Cannabinoid Receptor 2' and Monomerid = 50258570
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50258570(CHEMBL466223 | N-(4-Methylcyclohexyl)-1-(2-morphol...)
Affinity DataKi:  1.90nMAssay Description:HEK293DHEK293iHEK293sHEK293pHEK293lHEK293aHEK293cHEK293eHEK293mHEK293eHEK293nHEK293tHEK293 HEK293oHEK293fHEK293 HEK293[HEK2933HEK293HHEK293]HEK293CHE...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50258570(CHEMBL466223 | N-(4-Methylcyclohexyl)-1-(2-morphol...)
Affinity DataKi:  1.90nMAssay Description:Displacement of [3H]CP-55940 from human recombinant CB2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50258570(CHEMBL466223 | N-(4-Methylcyclohexyl)-1-(2-morphol...)
Affinity DataIC50:  210nMAssay Description:HEK293DHEK293iHEK293sHEK293pHEK293lHEK293aHEK293cHEK293eHEK293mHEK293eHEK293nHEK293tHEK293 HEK293oHEK293fHEK293 HEK293[HEK2933HEK293HHEK293]HEK293CHE...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50258570(CHEMBL466223 | N-(4-Methylcyclohexyl)-1-(2-morphol...)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human recombinant CB2R expressed in U2OS cells assessed as beta-arrestin-GFP binding to receptor after 25 mins by fluorescent mic...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50258570(CHEMBL466223 | N-(4-Methylcyclohexyl)-1-(2-morphol...)
Affinity DataEC50:  28nMAssay Description:Agonist activity at human recombinant CB2R expressed in WIN-55212-stimulated U2OS cells assessed as reduction in forskolin-mediated cAMP level after ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed