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Found 1 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M3' and Monomerid = 50267811
TargetMuscarinic acetylcholine receptor M3(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50267811(4-(Hydroxy{bis[4-(methyloxy)phenyl]}methyl)-1-{2-[...)
Affinity DataIC50:  3.60E+4nMAssay Description:Antagonist activity at human cloned muscarinic M3 receptor expressed in CHO cells assessed as inhibition of acetylcholine-induced calcium mobilizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed