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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 Receptor' and Monomerid = 50268508
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50268508((5-fluoro-6-(1-isopropylpiperidin-4-yloxy)-1H-indo...)
Affinity DataKi:  366nMAssay Description:Displacement of [3H](R)-alpha-methylhistamine from human recombinant histamine H3 receptor expressed in CHO cells by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50268508((5-fluoro-6-(1-isopropylpiperidin-4-yloxy)-1H-indo...)
Affinity DataEC50:  112nMAssay Description:Inverse agonist activity at human histamine H3 receptor expressed in CHO cells by GTPgamma[35S] binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed