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Found 2 Enz. Inhib. hit(s) with Target = 'Thromboxane A2 receptor' and Monomerid = 50277668
TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50277668((R)-2-(9-(3,4-dichlorophenylthio)-1-isopropyl-7,8-...)
Affinity DataKi:  935nMAssay Description:Displacement of radioligand from human recombinant TP receptor expressed in HEK293 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThromboxane A2 receptor(Homo sapiens (Human))
Merck Frosst Centre For Therapeutic Research

Curated by ChEMBL
LigandPNGBDBM50277668((R)-2-(9-(3,4-dichlorophenylthio)-1-isopropyl-7,8-...)
Affinity DataIC50:  4.04E+3nMAssay Description:Antagonist activity at TP1 in human platelet-rich plasma assessed as inhibition of U44619-induced platelet aggregationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed