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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Monomerid = 50280563
LigandPNGBDBM50280563(1-Aza-bicyclo[2.2.1]heptan-3-one O-(4-methoxy-but-...)
Affinity DataIC50:  55nMAssay Description:Compound was evaluated for inhibition of [3H]cis-methyldioxolane binding to label agonist sites (RCMD) in rat neocortexMore data for this Ligand-Target Pair
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TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50280563(1-Aza-bicyclo[2.2.1]heptan-3-one O-(4-methoxy-but-...)
Affinity DataIC50:  4.24E+4nMAssay Description:Inhibitory activity against human Muscarinic acetylcholine receptor M1 using [3H]-quinuclidinyl benzilate to label antagonist site (RQNB) in CHO cell...More data for this Ligand-Target Pair
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