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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Plasmin' and Monomerid = 50289373   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Plasminogen


(Homo sapiens (Human))
BDBM50289373
PNG
(2-(4-Chloro-benzenesulfonylamino)-N-[(R)-1-(piperi...)
Show SMILES Clc1ccc(cc1)S(=O)(=O)NCC(=O)N[C@H](CCNc1ccncc1)C(=O)N1CCCCC1
Show InChI InChI=1S/C22H28ClN5O4S/c23-17-4-6-19(7-5-17)33(31,32)26-16-21(29)27-20(22(30)28-14-2-1-3-15-28)10-13-25-18-8-11-24-12-9-18/h4-9,11-12,20,26H,1-3,10,13-16H2,(H,24,25)(H,27,29)/t20-/m1/s1
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Similars

Article
>5.00E+5n/an/an/an/an/an/a7.5n/a



TBA

Curated by ChEMBL


Assay Description
Tested for the Inhibition of the catalytic activity of human plasmin at 25 degree C and pH 7.5.


Bioorg Med Chem Lett 7: 1283-1288 (1997)


Article DOI: 10.1016/S0960-894X(97)00210-2
BindingDB Entry DOI: 10.7270/Q29W0FZ9
More data for this
Ligand-Target Pair