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Found 2 Enz. Inhib. hit(s) with Target = 'ATP-Binding Cassette Transporter ABCG2' and Monomerid = 50293013
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50293013(CHEMBL455275 | Methyl 4-((4-(2-(6,7-dimethoxy-1,2,...)
Affinity DataIC50:  172nMAssay Description:Inhibition of ABCG2 expressed in human MCF7/Topo cells by Hoechst microplate assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universidad Nacional De Colombia

Curated by ChEMBL
LigandPNGBDBM50293013(CHEMBL455275 | Methyl 4-((4-(2-(6,7-dimethoxy-1,2,...)
Affinity DataIC50:  179nMAssay Description:Inhibition of ABCG2 overexpressed in human MCF7/Topo cells by flow cytometric-based mitoxantrone efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed