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Found 3 Enz. Inhib. hit(s) with Target = 'Cruzipain' and Monomerid = 50295106
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295106(5-(2-Amino-phenyl)-[1,3,4]oxadiazole-2-carboxylic ...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain preincubated for 5 mins before substrate additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295106(5-(2-Amino-phenyl)-[1,3,4]oxadiazole-2-carboxylic ...)
Affinity DataIC50: >2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain preincubated for 5 mins before substrate addition in presence of 0.01% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCruzipain(Trypanosoma cruzi)
University Of California

Curated by ChEMBL
LigandPNGBDBM50295106(5-(2-Amino-phenyl)-[1,3,4]oxadiazole-2-carboxylic ...)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Trypanosoma cruzi cruzain preincubated for 5 mins before substrate addition in presence of 0.001% Triton X-100More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed