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Found 1 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50295635
TargetGlucocorticoid receptor(Homo sapiens (Human))
Johnson And Johnson Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50295635((1R,3S,3aR,3bS,10R)-1-Ethynyl-1-hydroxy-10-(4-meth...)
Affinity DataIC50:  110nMAssay Description:Antagonist activity at glucocorticoid receptor in human A549 cells assessed as inhibition of corticoid-induced transcription after 16 hrs by glucocor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed