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Found 1 hit Enz. Inhib. hit(s) with Target = 'Telomerase reverse transcriptase' and Monomerid = 50298386   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Telomerase reverse transcriptase


(Homo sapiens (Human))
BDBM50298386
PNG
(4,5-Bis(aminomethyl)acridine dihydrochloride salt ...)
Show SMILES NCc1cccc2cc3cccc(CN)c3nc12
Show InChI InChI=1S/C15H15N3/c16-8-12-5-1-3-10-7-11-4-2-6-13(9-17)15(11)18-14(10)12/h1-7H,8-9,16-17H2
PDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a>3.00E+4n/an/an/an/an/an/a



Universit£ de Reims Champagne-Ardenne

Curated by ChEMBL


Assay Description
Inhibition of human telomerase in A549 cells by TRAP assay


Eur J Med Chem 44: 3880-8 (2009)


Article DOI: 10.1016/j.ejmech.2009.04.021
BindingDB Entry DOI: 10.7270/Q2W37WDH
More data for this
Ligand-Target Pair