Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Monomerid = 50311793
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  790nMAssay Description:Agonist activity at PPARalpha receptor expressed in HEK293 cells cotransfected with GAL4 by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  790nMAssay Description:Agonist activity at PPARalphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
The University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50311793(4'-butoxy-3'-((2-fluoro-4-(trifluoromethyl)benzami...)
Affinity DataEC50:  790nMAssay Description:Partial agonist activity at human recombinant PPARalpha LBD expressed in HEK293 cells cotransfected with Gal4 assessed as beta-galactosidase activity...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed