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Found 2 Enz. Inhib. hit(s) with Target = 'Cathepsin S' and Monomerid = 50314235
TargetCathepsin S(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50314235(CHEMBL1090995 | rac-2-(5-(1-(3-(4-(3-methyl-1,2,4-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human recombinant cathepsin S expressed in baculovirus expression sytem after 15 mins by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCathepsin S(Homo sapiens (Human))
Johnson & Johnson Pharmaceutical Research & Development

Curated by ChEMBL
LigandPNGBDBM50314235(CHEMBL1090995 | rac-2-(5-(1-(3-(4-(3-methyl-1,2,4-...)
Affinity DataIC50:  3.46E+3nMAssay Description:Inhibition of cathepsin S in human JY cells assessed as accumulation of invariant chain p10li after 24 hrs by Western blot analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed