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Found 1 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M5' and Monomerid = 50314597
TargetMuscarinic acetylcholine receptor M5(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50314597(CHEMBL1090097 | N-(3-chloro-4-(4-ethylpiperazin-1-...)
Affinity DataIC50:  4.10E+3nMAssay Description:Antagonist activity at human muscarinic M5 receptor expressed in CHO-K1 cells assessed as inhibition of acetylcholine-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed