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Found 1 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Monomerid = 50314599
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50314599(CHEMBL1093933 | N-(3-chloro-4-(4-ethylpiperazin-1-...)
Affinity DataIC50:  4.70E+3nMAssay Description:Antagonist activity at human muscarinic M1 receptor expressed in CHO-K1 cells assessed as inhibition of acetylcholine-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed