Found 7 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Monomerid = 50318462
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Antagonist activity at human TRPA1 channel assessed as inhibition of trinitrophenol-induced responseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Antagonist activity at human TRPA1 channel assessed as inhibition of hypertonic solution of 400 mOsm-induced responseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataIC50: 850nMAssay Description:Antagonist activity at human TRPA1 channel assessed as inhibition of URB597-induced intracellular calcium influxMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human TRPA1 channel assessed as inhibition of 4-hydroxy-2-nonenal-induced responseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human TRPA1 channel assessed as inhibition of allyl isothiocyanate-induced intracellular calcium influxMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at human TRPA1 channel assessed as inhibition of cynnamaldehyde-induced responseMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
Ferrara University
Curated by ChEMBL
Ferrara University
Curated by ChEMBL
Affinity DataEC50: 4nMAssay Description:Agonist activity at TRPA1 channel in rat DRG neurons assessed as increase in intracellular calcium influxMore data for this Ligand-Target Pair