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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50318934
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50318934(2-(3-(4-cyanophenoxy)-2,4-dicyclopropyl-1H-pyrrol-...)
Affinity DataIC50:  47nMAssay Description:Antagonist activity at human recombinant progesterone receptor expressed in CHO-MMTV-beta-lactamase cells assessed as inhibition of progesterone-indu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50318934(2-(3-(4-cyanophenoxy)-2,4-dicyclopropyl-1H-pyrrol-...)
Affinity DataIC50:  4.00E+4nMAssay Description:Antagonist activity at progesterone receptor in human T47D cells by alkaline phosphatase releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed