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Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 Receptor' and Monomerid = 50319515
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50319515((R)-2,6-dimethyl-5-(6-(2-(2-methylpyrrolidin-1-yl)...)
Affinity DataKi:  0.980nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from human cloned histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50319515((R)-2,6-dimethyl-5-(6-(2-(2-methylpyrrolidin-1-yl)...)
Affinity DataKi:  1nMAssay Description:Displacement of [125I]Iodoproxyfan from human recombinant histamine H3 receptor by Competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50319515((R)-2,6-dimethyl-5-(6-(2-(2-methylpyrrolidin-1-yl)...)
Affinity DataKi:  5.5nMAssay Description:Displacement of [3H]-N-alpha-methylhistamine from rat cloned histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed