Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Peroxisome Proliferator-Activated Receptor gamma' and Monomerid = 50320886
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Universidade Federal De Pernambuco

Curated by ChEMBL
LigandPNGBDBM50320886(3-(2-Bromo-benzyl)-5-(4-methanesulfonyl-benzyliden...)
Affinity DataKi:  7.30E+3nMAssay Description:Displacement of [3H]rosiglitazone from human PPARgamma ligand binding domain expressed in Escherichia coli BL21 after 12 hrs by liquid scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed