Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase ABL' and Monomerid = 50323777
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50323777(CHEMBL1214141 | N-(4-Methyl-3-(1-methyl-7-(6-methy...)
Affinity DataIC50:  1.25nMAssay Description:Inhibition of wild type Bcr-AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBreakpoint cluster region protein/Tyrosine-protein kinase ABL1(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50323777(CHEMBL1214141 | N-(4-Methyl-3-(1-methyl-7-(6-methy...)
Affinity DataIC50:  1.25nMAssay Description:Inhibition of wild type Bcr-Abl using Tyr2 peptide as substrate after 2 hrs by FRET-based Z'-Lyte assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Harvard Medical School

Curated by ChEMBL
LigandPNGBDBM50323777(CHEMBL1214141 | N-(4-Methyl-3-(1-methyl-7-(6-methy...)
Affinity DataIC50:  133nMAssay Description:Inhibition of c-AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed