Compile Data Set for Download or QSAR
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Found 1 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50324116
TargetProgesterone receptor(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50324116((R)-Methyl 2-((1H-Tetrazol-1-yl)methyl)-4-(2-chlor...)
Affinity DataIC50:  7.20E+3nMAssay Description:Antagonist activity at progesterone receptor LBD expressed in human HUH7 cells coexpressing GAL4 by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed