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Found 2 Enz. Inhib. hit(s) with Target = 'Caspase-3' and Monomerid = 50326094
TargetCaspase-3(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50326094((S)-3-((S)-2-(benzyloxycarbonylamino)-3-methylbuta...)
Affinity DataIC50:  3.53E+4nMAssay Description:Inhibition of human recombinant caspase-3 expressed in Saccharomyces cerevisiae CG379 assessed as growth stimulation after 2 daysMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCaspase-3(Homo sapiens (Human))
University Of Lisbon

Curated by ChEMBL
LigandPNGBDBM50326094((S)-3-((S)-2-(benzyloxycarbonylamino)-3-methylbuta...)
Affinity DataIC50:  1.33E+5nMAssay Description:Inhibition of human recombinant caspase 3 assessed as fluorescent 7-amido-4-methylcoumarin releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed