BindingDB logo
myBDB logout
Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase SRC' and Monomerid = 50329876   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Proto-oncogene tyrosine-protein kinase Src


(Homo sapiens (Human))
BDBM50329876
PNG
(4-(5-(6-oxo-1,6-dihydropyridin-3-yl)oxazol-2-ylami...)
Show SMILES NS(=O)(=O)c1ccc(Nc2ncc(o2)-c2ccc(=O)[nH]c2)cc1
Show InChI InChI=1S/C14H12N4O4S/c15-23(20,21)11-4-2-10(3-5-11)18-14-17-8-12(22-14)9-1-6-13(19)16-7-9/h1-8H,(H,16,19)(H,17,18)(H2,15,20,21)
PDB
MMDB

KEGG

UniProtKB/SwissProt

B.MOAD
DrugBank
GoogleScholar
AffyNet 
CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/a 8.20E+3n/an/an/an/an/an/a



Ansaris

Curated by ChEMBL


Assay Description
Inhibition of c-SRC by Hot Spot filtration binding assay


Bioorg Med Chem Lett 20: 6394-9 (2010)


Article DOI: 10.1016/j.bmcl.2010.09.088
BindingDB Entry DOI: 10.7270/Q2NP24NB
More data for this
Ligand-Target Pair