Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'DNA Gyrase Subunit B' and Monomerid = 50330306
TargetDNA gyrase subunit B(Escherichia coli (strain K12))
UniversitäT TüBingen

Curated by ChEMBL
LigandPNGBDBM50330306((3R,4S,5R,6R)-6-(3-(4-amino-3-methylbenzamido)-4-h...)
Affinity DataIC50:  44nMAssay Description:Inhibition of Escherichia coli JM109 DNA gyrase subunit B assessed as DNA triple helix formation by supercoiling assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit B(Escherichia coli (strain K12))
UniversitäT TüBingen

Curated by ChEMBL
LigandPNGBDBM50330306((3R,4S,5R,6R)-6-(3-(4-amino-3-methylbenzamido)-4-h...)
Affinity DataIC50:  152nMAssay Description:Inhibition of Escherichia coli JM109 DNA gyrase subunit B assessed as ATP hydrolysis by ATPase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed