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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 2' and Monomerid = 50331744   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Metabotropic glutamate receptor 2


(Homo sapiens (Human))
BDBM50331744
PNG
((S)-1-(2-amino-2-carboxyethyl)-1H-1,2,3-triazole-4...)
Show SMILES N[C@@H](Cn1cc(nn1)C(O)=O)C(O)=O
Show InChI InChI=1S/C6H8N4O4/c7-3(5(11)12)1-10-2-4(6(13)14)8-9-10/h2-3H,1,7H2,(H,11,12)(H,13,14)/t3-/m0/s1
PDB

UniProtKB/SwissProt

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CHEMBL
PC cid
PC sid
UniChem
Article
PubMed
n/an/an/an/a>1.00E+5n/an/an/an/a



The University of Adelaide

Curated by ChEMBL


Assay Description
Binding affinity at mGluR2 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP production after 10 mins


Bioorg Med Chem Lett 20: 7512-5 (2010)


Article DOI: 10.1016/j.bmcl.2010.09.139
BindingDB Entry DOI: 10.7270/Q2K64J94
More data for this
Ligand-Target Pair