Affinity DataKi: 0.00300nMAssay Description:Binding affinity to dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.220nMAssay Description:Binding affinity to dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 7.93nMAssay Description:Binding affinity at NETMore data for this Ligand-Target Pair
Affinity DataKi: 8.29nMAssay Description:Binding affinity at NETMore data for this Ligand-Target Pair
Affinity DataKi: 10.8nMAssay Description:Binding affinity at NETMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [125I]PE2I from rat DATMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Displacement of [125I]PE2I from rat DATMore data for this Ligand-Target Pair
Affinity DataIC50: 3.40nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of human PARP1More data for this Ligand-Target Pair
Affinity DataKd: 200nMAssay Description:Binding affinity to human PARP1More data for this Ligand-Target Pair
Affinity DataKd: 19nMAssay Description:Binding affinity to human PARP1 by isothermal titration colorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 110nMAssay Description:Binding affinity to human PARP1 by isothermal titration colorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 150nMAssay Description:Binding affinity to human PARP1 by isothermal titration colorimetryMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP3 [R100H](Homo sapiens (Human))
Institutet
Curated by ChEMBL
Institutet
Curated by ChEMBL
Affinity DataKd: 70nMAssay Description:Binding affinity to human PARP3 PARP domain by isothermal titration colorimetryMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP3 [R100H](Homo sapiens (Human))
Institutet
Curated by ChEMBL
Institutet
Curated by ChEMBL
Affinity DataKd: 700nMAssay Description:Binding affinity to human PARP3 PARP domain by isothermal titration colorimetryMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP3 [R100H](Homo sapiens (Human))
Institutet
Curated by ChEMBL
Institutet
Curated by ChEMBL
Affinity DataKd: 2.00E+3nMAssay Description:Binding affinity to human PARP3 PARP domain by isothermal titration colorimetryMore data for this Ligand-Target Pair
TargetProtein mono-ADP-ribosyltransferase PARP3 [R100H](Homo sapiens (Human))
Institutet
Curated by ChEMBL
Institutet
Curated by ChEMBL
Affinity DataKd: >2.00E+3nMAssay Description:Binding affinity to human PARP3 PARP domain by isothermal titration colorimetryMore data for this Ligand-Target Pair
Affinity DataKd: 9.40E+4nMAssay Description:Binding affinity to human CBS by PLP fluorescence-based screening assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.0510nMAssay Description:Binding affinity of the radio labeled [3H]-5-Methyl-6-nitroquipazine compound against Serotonin transporter in rat frontal cortex homogenatesMore data for this Ligand-Target Pair
Affinity DataKd: 0.0510nMAssay Description:Binding affinity of the radio labeled [3H]-5-Methyl-6-nitroquipazine compound against Serotonin transporter in rat frontal cortex homogenatesMore data for this Ligand-Target Pair