Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50121649![]() (2-[({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | 0.0210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomes | J Med Chem 45: 5556-63 (2002) Article DOI: 10.1021/jm020336e BindingDB Entry DOI: 10.7270/Q2BR8SWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50194487![]() (3-[4'-(H-Dmt)-aminobutyl]-6-[3'-(H-Dmt)-aminopropy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fraction | Bioorg Med Chem Lett 16: 5793-6 (2006) Article DOI: 10.1016/j.bmcl.2006.08.079 BindingDB Entry DOI: 10.7270/Q26Q1WWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50179190![]() (2-(2-(((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0210 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin II from rat delta opioid receptor in brain P2 synaptosomes | J Med Chem 48: 8112-4 (2005) Article DOI: 10.1021/jm058259l BindingDB Entry DOI: 10.7270/Q24J0DQR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50266025![]() ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliary Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assay | J Med Chem 45: 713-20 (2002) Article DOI: 10.1021/jm010449i BindingDB Entry DOI: 10.7270/Q2639QFF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50266025![]() ((S)-2-((S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0310 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Brussels Curated by ChEMBL | Assay Description Binding affinity to delta opioid receptor | J Med Chem 49: 3990-3 (2006) Article DOI: 10.1021/jm0603264 BindingDB Entry DOI: 10.7270/Q2474BPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50027229![]() (CHEMBL2375157) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Brussels Curated by ChEMBL | Assay Description Binding affinity to delta opioid receptor | J Med Chem 49: 3990-3 (2006) Article DOI: 10.1021/jm0603264 BindingDB Entry DOI: 10.7270/Q2474BPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50179191![]() ((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin II from rat delta opioid receptor in brain P2 synaptosomes | J Med Chem 48: 8112-4 (2005) Article DOI: 10.1021/jm058259l BindingDB Entry DOI: 10.7270/Q24J0DQR | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50179191![]() ((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliary Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assay | J Med Chem 45: 713-20 (2002) Article DOI: 10.1021/jm010449i BindingDB Entry DOI: 10.7270/Q2639QFF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50179191![]() ((S)-N-((1H-benzo[d]imidazol-2-yl)methyl)-2-((S)-2-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0350 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomes | J Med Chem 45: 5556-63 (2002) Article DOI: 10.1021/jm020336e BindingDB Entry DOI: 10.7270/Q2BR8SWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50130611![]() (2-Amino-N-{4-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparation | J Med Chem 46: 3201-9 (2003) Article DOI: 10.1021/jm020459z BindingDB Entry DOI: 10.7270/Q28C9VMQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50157686![]() (5-[({5-[(2S)-2-({2-[(2S)-2-amino-3-(4-hydroxy-2,6-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem | Article PubMed | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliary Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from delta opioid receptor in rat brain synaptosomes P2 fraction | J Med Chem 47: 6541-6 (2004) Article DOI: 10.1021/jm040128h BindingDB Entry DOI: 10.7270/Q28W3CS2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50083160![]() ((S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0400 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement. | J Med Chem 42: 5010-9 (2000) Article DOI: 10.1021/jm990165m BindingDB Entry DOI: 10.7270/Q2VX0FQG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50272081![]() (2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliary Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assay | J Med Chem 45: 713-20 (2002) Article DOI: 10.1021/jm010449i BindingDB Entry DOI: 10.7270/Q2639QFF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50121648![]() (2-({2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | 0.0420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomes | J Med Chem 45: 5556-63 (2002) Article DOI: 10.1021/jm020336e BindingDB Entry DOI: 10.7270/Q2BR8SWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50221787![]() (CHEMBL3216418) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institutes of Environmental Health Sciences Curated by ChEMBL | Assay Description Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileum | J Med Chem 47: 2599-610 (2004) Article DOI: 10.1021/jm0304616 BindingDB Entry DOI: 10.7270/Q2RB755V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Delta-type opioid receptor (Homo sapiens (Human)) | BDBM50272081![]() (2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0420 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Brussels Curated by ChEMBL | Assay Description Binding affinity to delta opioid receptor | J Med Chem 49: 3990-3 (2006) Article DOI: 10.1021/jm0603264 BindingDB Entry DOI: 10.7270/Q2474BPW | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50212613![]() (CHEMBL266122 | Tyr-Pro-Dmp-Phe-NH2) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0440 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane | J Med Chem 50: 2753-66 (2007) Article DOI: 10.1021/jm061238m BindingDB Entry DOI: 10.7270/Q25B0264 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50049378![]() (1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0450 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1 | J Med Chem 39: 773-80 (1996) Article DOI: 10.1021/jm950490j BindingDB Entry DOI: 10.7270/Q2QV3KKJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50121645![]() (2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)pr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | 0.0470 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomes | J Med Chem 45: 5556-63 (2002) Article DOI: 10.1021/jm020336e BindingDB Entry DOI: 10.7270/Q2BR8SWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50130617![]() (2-Amino-N-{6-[2-amino-3-(4-hydroxy-2,6-dimethyl-ph...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0500 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Binding affinity for Opioid receptor mu 1 using [3H]-DAGO in rat brain P2 synaptosomal preparation | J Med Chem 46: 3201-9 (2003) Article DOI: 10.1021/jm020459z BindingDB Entry DOI: 10.7270/Q28C9VMQ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50194488![]() (6-[4'-(H-Dmt)-aminobutyl]-3-[3'-(H-Dmt)-aminopropy...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0510 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat synaptosomes P2 fraction | Bioorg Med Chem Lett 16: 5793-6 (2006) Article DOI: 10.1016/j.bmcl.2006.08.079 BindingDB Entry DOI: 10.7270/Q26Q1WWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50049377![]() (1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1 | J Med Chem 39: 773-80 (1996) Article DOI: 10.1021/jm950490j BindingDB Entry DOI: 10.7270/Q2QV3KKJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50199865![]() ((S)-N-((S)-1-((S)-1-amino-1-oxo-3-phenylpropan-2-y...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in rat brain P2 synaptosome | Bioorg Med Chem 15: 1237-51 (2007) Article DOI: 10.1016/j.bmc.2006.11.019 BindingDB Entry DOI: 10.7270/Q2348K1F | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50049376![]() (1-((S)-2-{(S)-2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0540 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Displacement of [3H]-DPDPE (0.63 nM) from Opioid receptor delta 1 | J Med Chem 39: 773-80 (1996) Article DOI: 10.1021/jm950490j BindingDB Entry DOI: 10.7270/Q2QV3KKJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50083154![]() ((S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0580 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement. | J Med Chem 42: 5010-9 (2000) Article DOI: 10.1021/jm990165m BindingDB Entry DOI: 10.7270/Q2VX0FQG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50157684![]() (CHEMBL2369958 | H-Dmt-Tic-Glu-NH2) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliary Curated by ChEMBL | Assay Description Displacement of [3H]DPDPE from delta opioid receptor in rat brain synaptosomes P2 fraction | J Med Chem 47: 6541-6 (2004) Article DOI: 10.1021/jm040128h BindingDB Entry DOI: 10.7270/Q28W3CS2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50178759![]() (1,6-bis-(N,N-dimethyl-Dmt-Tic-NH)hexane | CHEMBL37...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0600 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranes | J Med Chem 48: 8035-44 (2005) Article DOI: 10.1021/jm050377l BindingDB Entry DOI: 10.7270/Q2C53KD9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50121645![]() (2-[(2S)-2-amino-3-(4-hydroxy-2,6-dimethylphenyl)pr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | 0.0630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomes | J Med Chem 45: 5556-63 (2002) Article DOI: 10.1021/jm020336e BindingDB Entry DOI: 10.7270/Q2BR8SWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50159681![]() ((S)-1-[2-Amino-3-(2-ethyl-4-hydroxy-6-methyl-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0630 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to mu-Opioid receptor | J Med Chem 48: 586-92 (2005) Article DOI: 10.1021/jm049384k BindingDB Entry DOI: 10.7270/Q26T0M40 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50083169![]() ((S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0660 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement. | J Med Chem 42: 5010-9 (2000) Article DOI: 10.1021/jm990165m BindingDB Entry DOI: 10.7270/Q2VX0FQG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50108919![]() (2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | 0.0670 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliary Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 using rat brain receptor (P2 synaptosome) assay | J Med Chem 45: 713-20 (2002) Article DOI: 10.1021/jm010449i BindingDB Entry DOI: 10.7270/Q2639QFF | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50108919![]() (2-[2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-propi...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | PC cid PC sid UniChem Similars | Article PubMed | 0.0670 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Cagliari Curated by ChEMBL | Assay Description Inhibition of [3H]DPDPE binding to Opioid receptor delta 1 of rat brain P2 synaptosomes | J Med Chem 45: 5556-63 (2002) Article DOI: 10.1021/jm020336e BindingDB Entry DOI: 10.7270/Q2BR8SWH | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50212609![]() (CHEMBL228409 | Dmt-Pro-Dmp-Phe-NH2) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0690 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane | J Med Chem 50: 2753-66 (2007) Article DOI: 10.1021/jm061238m BindingDB Entry DOI: 10.7270/Q25B0264 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50001459![]() (3-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0700 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Tested for inhibition of amplification of electrically induced twitch in guinea pig ileum (GPI) | J Med Chem 36: 3748-56 (1994) Article DOI: 10.1021/jm00076a001 BindingDB Entry DOI: 10.7270/Q2D799HM | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50083160![]() ((S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0730 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by [3H]N,N-(Me)2-Dmt-Tic-OH displacement. | J Med Chem 42: 5010-9 (2000) Article DOI: 10.1021/jm990165m BindingDB Entry DOI: 10.7270/Q2VX0FQG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50060083![]() (2-({2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0755 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPE | J Med Chem 40: 3100-8 (1997) Article DOI: 10.1021/jm9607663 BindingDB Entry DOI: 10.7270/Q2TD9Z1N | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50083169![]() ((S)-2-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-pheny...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0800 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement. | J Med Chem 42: 5010-9 (2000) Article DOI: 10.1021/jm990165m BindingDB Entry DOI: 10.7270/Q2VX0FQG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50159684![]() ((S)-1-[2-Amino-3-(2,6-diethyl-4-hydroxy-phenyl)-pr...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0840 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to mu-Opioid receptor | J Med Chem 48: 586-92 (2005) Article DOI: 10.1021/jm049384k BindingDB Entry DOI: 10.7270/Q26T0M40 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50212619![]() (CHEMBL388800 | Dmt-Pro-Dmt-Phe-NH2) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0920 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane | J Med Chem 50: 2753-66 (2007) Article DOI: 10.1021/jm061238m BindingDB Entry DOI: 10.7270/Q25B0264 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50178757![]() (3-(Dmt-Tic-NH-butyl)-6-(Dmt-Tic-NH-propyl)-2-(1H)-...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0920 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranes | J Med Chem 48: 8035-44 (2005) Article DOI: 10.1021/jm050377l BindingDB Entry DOI: 10.7270/Q2C53KD9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50178761![]() (3,6-bis(Dmt-Tic-NH-ethyl)-2(1H)-pyrazinone | CHEMB...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.0950 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranes | J Med Chem 48: 8035-44 (2005) Article DOI: 10.1021/jm050377l BindingDB Entry DOI: 10.7270/Q2C53KD9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50178756![]() (3-(Dmt-Tic-NH-ethyl)-6-(Dmt-Tic-NH-butyl)-2-(1H)-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.107 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]deltorphin-II from delta opioid receptor in rat brain synaptosomal membranes | J Med Chem 48: 8035-44 (2005) Article DOI: 10.1021/jm050377l BindingDB Entry DOI: 10.7270/Q2C53KD9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50083167![]() ((S)-2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimeth...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity at Opioid receptor delta 1 from rat brain synaptosomal preparations by H-Dmt-Tic-OH displacement. | J Med Chem 42: 5010-9 (2000) Article DOI: 10.1021/jm990165m BindingDB Entry DOI: 10.7270/Q2VX0FQG | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50059366![]() (((S)-2-{(S)-2-[2-((S)-2-{(R)-2-[(S)-2-Amino-3-(4-h...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institute of Environmental Health Sciences Curated by ChEMBL | Assay Description Affinity of the compound was assessed using competitive binding assay labeled with [3H]-DPDPE (6.3 nM) for Opioid receptor delta 1 | J Med Chem 40: 2579-87 (1997) Article DOI: 10.1021/jm9700530 BindingDB Entry DOI: 10.7270/Q25M64T2 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50212616![]() (CHEMBL389949 | Dmt-Pro-3,5Dmp-Phe-NH2) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosome membrane | J Med Chem 50: 2753-66 (2007) Article DOI: 10.1021/jm061238m BindingDB Entry DOI: 10.7270/Q25B0264 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50149389![]() (1-[(S)-2-Amino-3-(4-hydroxy-2,6-dimethyl-phenyl)-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.110 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Binding affinity against rat brain Opioid receptor mu 1 using [3H]-DAMGO radioligand | J Med Chem 47: 3591-9 (2004) Article DOI: 10.1021/jm030649p BindingDB Entry DOI: 10.7270/Q2W095DJ | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50159680![]() ((S)-1-[2-Amino-3-(4-hydroxy-2,3,6-trimethyl-phenyl...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.111 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Kobe Gakuin University Curated by ChEMBL | Assay Description Inhibition of [3H]-DAMGO binding to mu-Opioid receptor | J Med Chem 48: 586-92 (2005) Article DOI: 10.1021/jm049384k BindingDB Entry DOI: 10.7270/Q26T0M40 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50221778![]() (CHEMBL3216392) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.114 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institutes of Environmental Health Sciences Curated by ChEMBL | Assay Description Compound was tested for binding affinity towards Opioid receptor mu 1 by displacing [3H]DAGO radioligand in rat brain P2 synaptosomes membranes. | J Med Chem 47: 2599-610 (2004) Article DOI: 10.1021/jm0304616 BindingDB Entry DOI: 10.7270/Q2RB755V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Nociceptin/mu opioid receptor (Rattus norvegicus (rat)) | BDBM50221781![]() (CHEMBL3215968) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.115 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
National Institutes of Environmental Health Sciences Curated by ChEMBL | Assay Description Compound was tested for Opioid receptor mu 1 agonism in isolated tissues from guinea pig ileum | J Med Chem 47: 2599-610 (2004) Article DOI: 10.1021/jm0304616 BindingDB Entry DOI: 10.7270/Q2RB755V | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Opioid receptors; mu & delta (Rattus norvegicus (rat)) | BDBM50060068![]() (2-[(S)-2-Dimethylamino-3-(4-hydroxy-2,6-dimethyl-p...) | PDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 0.118 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Ferrara Curated by ChEMBL | Assay Description Binding affinity for Opioid receptor delta 1 by displacement of [3H]- DPDPE | J Med Chem 40: 3100-8 (1997) Article DOI: 10.1021/jm9607663 BindingDB Entry DOI: 10.7270/Q2TD9Z1N | |||||||||||
More data for this Ligand-Target Pair |
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