Compile Data Set for Download or QSAR
maximum 50k data
Found 15 of ec50 for UniProtKB: P45983
TargetMitogen-activated protein kinase 10/8/9(Homo sapiens (Human))
National Clinical Research Center For Geriatrics

Curated by ChEMBL
LigandPNGBDBM86636(JNK-IN-11)
Affinity DataEC50:  8.60nMAssay Description:Inhibition of c-Jun phosphorylation in human A-375 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM60665(BDBM50249542 | US9145414, R406 | US9212178, R406)
Affinity DataEC50:  10nMAssay Description:Inhibition of JNK1 in OVA-challenged and IgE-sensitized cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 10/8/9(Homo sapiens (Human))
National Clinical Research Center For Geriatrics

Curated by ChEMBL
LigandPNGBDBM86636(JNK-IN-11)
Affinity DataEC50:  48nMAssay Description:Inhibition of c-Jun phosphorylation in human HeLa cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50352629(CHEMBL1822314)
Affinity DataEC50:  2.00E+3nMAssay Description:Inhibition of anisomycin-induced c-JUN phosphorylation in human HEK293T cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392984(CHEMBL2152384)
Affinity DataEC50:  3.30E+3nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392983(CHEMBL2152383)
Affinity DataEC50:  4.10E+3nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392990(CHEMBL2152390)
Affinity DataEC50:  4.10E+3nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392985(CHEMBL2152385)
Affinity DataEC50:  8.50E+3nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392988(CHEMBL2152388)
Affinity DataEC50:  9.00E+3nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392986(CHEMBL2152386)
Affinity DataEC50:  9.90E+3nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392982(CHEMBL2152382)
Affinity DataEC50:  1.01E+4nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50352629(CHEMBL1822314)
Affinity DataEC50:  1.40E+4nMAssay Description:Inhibition of TNFalpha-induced c-JUN phosphorylation in mouse B16-F10 cells by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392987(CHEMBL2152387)
Affinity DataEC50:  1.40E+4nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392989(CHEMBL2152389)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
Rigel

Curated by ChEMBL
LigandPNGBDBM50392992(CHEMBL2152392)
Affinity DataEC50:  2.19E+4nMAssay Description:Inhibition of JNK1-mediated c-jun phosphorylation in TNF-alpha stimulated human HK-2 cells after 30 mins by TR-FRET assayMore data for this Ligand-Target Pair