Found 9 hits of affinity data for UniProtKB/TrEMBL: P53582Target (Institution) | Ligand | Target Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | pH | Temp °C |
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | A311263
 ((2S,3R)-3-amino-5-(ethylsulfanyl)-2-hydroxy-N-[(1S...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| B.MOAD CHEBI CSLS MMDB PC cid PC sid PDB
| PubMed
| n/a | n/a | 370.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | bestatin-type inhibitor, 5
 ((2S,3S)-3-amino-2-hydroxy-4-[(2-methylpropyl)sulfa...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| CHEBI PC cid PC sid
| PubMed
| n/a | n/a | 2200.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | bestatin-type inhibitor, 8
 (N'-[(2S,3S)-3-amino-2-hydroxy-4-[(2-methylpropyl)s...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| CHEBI PC cid PC sid
| PubMed
| n/a | n/a | 8100.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | bestatin-type inhibitor, 6
 ((2S,3R)-3-amino-2-hydroxy-N-[(1S)-1-(naphthalen-1-...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| CHEBI PC cid PC sid
| PubMed
| n/a | n/a | 12000.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | bestatin-type inhibitor, 7
 (N'-[(2S,3R)-3-amino-5-(ethylsulfanyl)-2-hydroxypen...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| CHEBI PC cid PC sid
| PubMed
| n/a | n/a | 20000.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | A-357300
 (N'-[(2S,3R)-3-amino-2-hydroxy-5-(propan-2-ylsulfan...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| B.MOAD CHEBI CSLS MMDB PC cid PC sid PDB
| PubMed
| n/a | n/a | 57000.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | bestatin-type inhibitor, 1
 (ethyl (2S)-2-[(2S,3R)-3-amino-2-hydroxy-5-(methyls...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| PC cid PC sid
| PubMed
| n/a | n/a | 63000.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | bestatin-type inhibitor, 3
 (ethyl (2S)-2-[(2S,3S)-3-amino-2-hydroxy-4-[(2-meth...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| PC cid PC sid
| PubMed
| n/a | n/a | 66000.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|
Methionine Aminopeptidase Type 1 (MetAP1)
Homo sapiens (human) | bestatin-type inhibitor, 2
 (ethyl (2S)-2-[(2S,3R)-3-amino-5-(ethylsulfanyl)-2-...) | B.MOAD GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL
| PC cid PC sid
| PubMed
| n/a | n/a | 69000.0 | n/a | n/a | 7.4 | 22 |
Abbott Laboratories
|
Cancer Res. 63: 7861-9 (2003)
|