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Found 18 of ic50 for UniProtKB: P0A079
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17871((1S)-1-[5-(benzylsulfanyl)-4H-1,2,4-triazol-3-yl]-...)
Affinity DataIC50:  43.7nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17870(1,2,4-triazole derivative. | 5-(benzylsulfanyl)-4H...)
Affinity DataIC50:  599nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17869((3S)-3-amino-1-(cyclopropylamino)heptane-2,2-diol ...)
Affinity DataIC50:  7.00E+3nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497527(CHEMBL3337741)
Affinity DataIC50:  7.00E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497528(CHEMBL3337742)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497533(CHEMBL3337746)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497517(CHEMBL3337739)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17868((2S)-2-amino-4-(methylsulfanyl)-1-(pyridin-2-yl)bu...)
Affinity DataIC50:  1.60E+4nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497525(CHEMBL3337744)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497519(CHEMBL3337745)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497532(CHEMBL3337751)
Affinity DataIC50:  1.89E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17867((2S)-2-amino-4-(methylsulfanyl)-1-(1,3-thiazol-2-y...)
Affinity DataIC50:  1.90E+4nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497523(CHEMBL3337736)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497530(CHEMBL3337638)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497518(CHEMBL3337738)
Affinity DataIC50:  3.20E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497529(CHEMBL3337743)
Affinity DataIC50:  4.21E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM50497526(CHEMBL3337737)
Affinity DataIC50:  4.60E+4nMAssay Description:Inhibition of N-terminal poly-His-tagged Staphylococcus aureus COL MetAP expressed in Escherichia coli BL21(DE3) incubated for 30 mins before MGMM su...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMethionine aminopeptidase(Staphylococcus aureus)
Morphochem

LigandPNGBDBM17872(1,2,4-triazole derivative. | 3-(benzylsulfanyl)-4-...)
Affinity DataIC50: >1.00E+5nMpH: 7.5 T: 2°CAssay Description:The MetAP reaction with Co2+ as a cofactor is coupled to a prolyl aminopeptidase (ProAP) using Met-Pro-p-nitroanilide as substrate. MetAP-catalyzed c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed