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Found 5 of ec50 for UniProtKB: P05412
TargetTranscription factor Jun(Homo sapiens (Human))
NCI-Frederick

Curated by ChEMBL
LigandPNGBDBM50349194(GLAUCARUBINONE | NSC-14975)
Affinity DataEC50:  130nMAssay Description:Inhibition of TPA-induced AP-1 activity expressed in human HEK293T cells treated 1 hr before TPA challenge measured after 18 hrs by FRET based beta-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
NCI-Frederick

Curated by ChEMBL
LigandPNGBDBM50349193(CHEMBL1807644)
Affinity DataEC50:  130nMAssay Description:Inhibition of AP-1 (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
NCI-Frederick

Curated by ChEMBL
LigandPNGBDBM15913(2-pyridinecarboxamide deriv. 8c | 4-Amino-5-cyano-...)
Affinity DataEC50:  318nMAssay Description:Inhibition of c-Jun phosphorylation in HepG2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
NCI-Frederick

Curated by ChEMBL
LigandPNGBDBM50349193(CHEMBL1807644)
Affinity DataEC50:  1.49E+3nMAssay Description:Inhibition of TPA-induced AP-1 activity expressed in human HEK293T cells treated 1 hr before TPA challenge measured after 18 hrs by FRET based beta-l...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTranscription factor Jun(Homo sapiens (Human))
NCI-Frederick

Curated by ChEMBL
LigandPNGBDBM50349194(GLAUCARUBINONE | NSC-14975)
Affinity DataEC50:  1.49E+3nMAssay Description:Inhibition of AP-1 (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed