PrimarySearch_ki

PrimarySearch_ki

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Found 2 hits affinity hit(s) for enzyme = Dihydrofolate Reductase (DHFR) with UniProtKB: P0A017
Target (Institution)	Ligand	Target Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	pH	Temp °C
Dihydrofolate Reductase (DHFR) Staphylococcus aureus	Trimethoprim (5-[(3,4,5-trimethoxyphenyl)methyl]pyrimidine-2,4-d...)	GoogleScholar PDB UniProtKB/SwissProt UniProtKB/TrEMBL	B.MOAD CSLS DrugBank PDB PubChem	PubMed	n/a	n/a	7.0	n/a	n/a	7	30
GSK		GoogleScholar PDB UniProtKB/SwissProt UniProtKB/TrEMBL	B.MOAD CSLS DrugBank PDB PubChem	PubMed	Bioorg Med Chem Lett. 13: 4217-21 (2003)
Dihydrofolate Reductase (DHFR) Staphylococcus aureus	Iclaprim (5-[(2-cyclopropyl-7,8-dimethoxy-2H-chromen-5-yl)me...)	GoogleScholar PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PubChem	PubMed	n/a	n/a	7.0	n/a	n/a	7	30
GSK		GoogleScholar PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PubChem	PubMed	Bioorg Med Chem Lett. 13: 4217-21 (2003)

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