PrimarySearch_ki

PrimarySearch_ki

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Found 4 hits affinity hit(s) for enzyme = tRNA synthetase (TyrRS) with UniProtKB: A5ITQ1
Target (Institution)	Ligand	Target Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	pH	Temp °C
tRNA synthetase (TyrRS) Staphylococcus aureus	SB-243545 (butyl (2S)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)prop...)	B.MOAD GoogleScholar MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PDB PubChem	PDB PubMed	n/a	n/a	0.2	n/a	n/a	7.9	37
GSK			CSLS PDB PubChem	PDB PubMed	Protein Sci. 10: 2008-16 (2001)
tRNA synthetase (TyrRS) Staphylococcus aureus	SB-219383 ((2S)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamid...)	B.MOAD GoogleScholar MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PDB PubChem	PDB PubMed	n/a	n/a	1.0	n/a	n/a	7.9	37
GSK			CSLS PDB PubChem	PDB PubMed	Protein Sci. 10: 2008-16 (2001)
tRNA synthetase (TyrRS) Staphylococcus aureus	SB-239629 ((2S)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamid...)	B.MOAD GoogleScholar MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PDB PubChem	PDB PubMed	n/a	n/a	3.0	n/a	n/a	7.9	37
GSK			CSLS PDB PubChem	PDB PubMed	Protein Sci. 10: 2008-16 (2001)
tRNA synthetase (TyrRS) Staphylococcus aureus	SB-284485 ((2S)-2-[(2S)-2-amino-3-(4-hydroxyphenyl)propanamid...)	B.MOAD GoogleScholar MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	B.MOAD CSLS PDB PubChem	B.MOAD PDB PubMed	n/a	n/a	4.0	n/a	n/a	7.9	37
GSK			B.MOAD CSLS PDB PubChem	B.MOAD PDB PubMed	Protein Sci. 10: 2008-16 (2001)

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Change energy unit to: kcal/mole