Compile Data Set for Download or QSAR
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Found 4 of ic50 for UniProtKB: P03406
TargetProtein Nef/Tyrosine-protein kinase HCK(Homo sapiens (Human))
University Of Pittsburgh

LigandPNGBDBM36545(DFP-4APF | diphenylfuropyrimidine-4-aminopropylfur...)
Affinity DataIC50:  2.00E+3nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Nef/Tyrosine-protein kinase HCK(Homo sapiens (Human))
University Of Pittsburgh

LigandPNGBDBM14807(3-(5,6-Diphenyl-furo[2,3-d]pyrimidin-4-ylamino)-pr...)
Affinity DataIC50:  5.10E+3nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Nef/Tyrosine-protein kinase HCK(Homo sapiens (Human))
University Of Pittsburgh

LigandPNGBDBM36544(DFP-4AB | Diphenylfuropyrimidine-4-aminobutanol)
Affinity DataIC50:  1.60E+4nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein Nef/Tyrosine-protein kinase HCK(Homo sapiens (Human))
University Of Pittsburgh

LigandPNGBDBM14806(5,6-Diphenyl-furo[2,3-d]pyrimidin-4 -ylamine | 5,6...)
Affinity DataIC50: >3.00E+4nMT: 2°CAssay Description:In vitro kinase activity of Nef-Hck complex and Hck alone using Z'-lyte kinase assay system and Tyr2 peptide substrate from Invitrogen.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed