Compile Data Set for Download or QSAR
maximum 50k data
Found 12 of ic50 for UniProtKB: P08962
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212272((R)-(4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]p...)
Affinity DataIC50:  33nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212270(6-(6-amino-5-methylpyrazin-2-yl)-N-(4-(4-(oxetan-3...)
Affinity DataIC50:  51nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212271(6-(6-aminopyrazin-2-yl)-N-(4-(4-(oxetan-3-yl)piper...)
Affinity DataIC50:  80nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM324284((R)-1-(tert-butyl)-N-(8-(2-((1-methyl-1H-pyrazol-4...)
Affinity DataIC50:  82nMAssay Description:Inhibition of CD63 (unknown origin) assessed as FcepsilonR induced basophil activationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212277(US11517570, Example Kn.-1: | US9290505, 6-(5-amino...)
Affinity DataIC50:  101nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212274(2-(5-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]pyrazi...)
Affinity DataIC50:  120nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212275(2-((4-(4-((6-(6-aminopyrazin-2-yl)imidazo[1,2-a]py...)
Affinity DataIC50:  128nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212273(6-(6-aminopyrazin-2-yl)-5-methyl-N-(4-(4-(oxetan-3...)
Affinity DataIC50:  157nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212276(2-(5-((6-(6-amino-5-methylpyrazin-2-yl)imidazo[1,2...)
Affinity DataIC50:  167nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212279(US11517570, Example Kn.-3: | US9290505, 6-(5-amino...)
Affinity DataIC50:  250nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212280(US11517570, Example Kn.-4: | US9290505, 6-(6-amino...)
Affinity DataIC50:  734nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetCD63 antigen(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM212278(US11517570, Example Kn.-2: | US9290505, 6-(3-amino...)
Affinity DataIC50:  809nMpH: 7.0Assay Description:Syk activity was measured using KinEASE (Cisbio), a time-resolved fluorescence resonance energy transfer (TR-FRET) immunoassay. In this assay, Syk-ca...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent