Compile Data Set for Download or QSAR
maximum 50k data
Found 603 of ic50 for Urease
having polymerids = 2721,5036,5908,9274,9993 and
complexids = 211,212
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50532145(CHEMBL1549559)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of jack bean urease assessed as reduction in ammonia production using urea as substrate after 15 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253257(CHEMBL4100084)
Affinity DataIC50:  50nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178021((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  58nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253269(CHEMBL4092986)
Affinity DataIC50:  60nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178020((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  64nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178016((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  72nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152597(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-nitrophenyl...)
Affinity DataIC50:  77nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178019((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  81nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178017((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  83nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178022((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  83nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178014((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  87nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178015((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  87nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152587(2-(1-(Benzofuran-2-yl)ethylidene)-N-phenylhydrazin...)
Affinity DataIC50:  89nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178013((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  96nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50356190(CHEMBL193474)
Affinity DataIC50:  102nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152600(2-(1-(Benzofuran-2-yl)ethylidene)-N-(3-methoxyphen...)
Affinity DataIC50:  102nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50123230(CHEMBL3622691)
Affinity DataIC50:  120nMAssay Description:Inhibition of jack beans urease assessed as hydrolysis of urea into ammonia preincubated for 10 mins followed by urea addition measured after 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50356195(CHEMBL241902)
Affinity DataIC50:  127nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM110170(Ethyl 4-[3-(3,4-dimethoxybenzoyl)thioureido]benzoa...)
Affinity DataIC50:  130nMpH: 8.2 T: 2°CAssay Description:The assay mixture contained 40 µL of buffer (0.01 M LiCl2, 1 mM EDTA, 0.01M K2HPO4, pH 8.2) containing 100 mM urea, 10 µL of enzyme (5U/mL)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253270(CHEMBL4071196)
Affinity DataIC50:  140nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50452584(CHEMBL4208211)
Affinity DataIC50:  140nMAssay Description:Inhibition of jack bean urease assessed as reduction in ammonia production using urea as substrate after 15 mins by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253275(CHEMBL4092021)
Affinity DataIC50:  150nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50123347(CHEMBL3622680)
Affinity DataIC50:  150nMAssay Description:Inhibition of jack beans urease assessed as hydrolysis of urea into ammonia preincubated for 10 mins followed by urea addition measured after 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50123229(CHEMBL3622693)
Affinity DataIC50:  160nMAssay Description:Inhibition of jack beans urease assessed as hydrolysis of urea into ammonia preincubated for 10 mins followed by urea addition measured after 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253254(CHEMBL4070510)
Affinity DataIC50:  170nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253258(CHEMBL4103174)
Affinity DataIC50:  170nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50356192(CHEMBL241894)
Affinity DataIC50:  177nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152591(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-fluoropheny...)
Affinity DataIC50:  177nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152598(2-(1-(Benzofuran-2-yl)ethylidene)-N-(4-nitrophenyl...)
Affinity DataIC50:  181nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM110169(Ethyl 4-[3-(4-methoxybenzoyl)thioureido]benzoate (...)
Affinity DataIC50:  210nMpH: 8.2 T: 2°CAssay Description:The assay mixture contained 40 µL of buffer (0.01 M LiCl2, 1 mM EDTA, 0.01M K2HPO4, pH 8.2) containing 100 mM urea, 10 µL of enzyme (5U/mL)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50356186(CHEMBL239452)
Affinity DataIC50:  215nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253271(CHEMBL4065321)
Affinity DataIC50:  220nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM53627(1-[[(E)-(5-oxidanyl-6-oxidanylidene-cyclohexa-2,4-...)
Affinity DataIC50:  220nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50356201(CHEMBL1910224)
Affinity DataIC50:  233nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM110165(Ethyl 4-[3-(3-chlorobenzoyl)thioureido]benzoate (1...)
Affinity DataIC50:  260nMpH: 8.2 T: 2°CAssay Description:The assay mixture contained 40 µL of buffer (0.01 M LiCl2, 1 mM EDTA, 0.01M K2HPO4, pH 8.2) containing 100 mM urea, 10 µL of enzyme (5U/mL)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50356197(CHEMBL1910221)
Affinity DataIC50:  263nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253273(CHEMBL4085244)
Affinity DataIC50:  280nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM110166(Ethyl 4-[3-(2,4-dichlorobenzoyl)thioureido]benzoat...)
Affinity DataIC50:  280nMpH: 8.2 T: 2°CAssay Description:The assay mixture contained 40 µL of buffer (0.01 M LiCl2, 1 mM EDTA, 0.01M K2HPO4, pH 8.2) containing 100 mM urea, 10 µL of enzyme (5U/mL)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM57806(1-[1-(1-benzofuran-2-yl)ethylideneamino]-3-(3-meth...)
Affinity DataIC50:  283nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253274(CHEMBL4100705)
Affinity DataIC50:  290nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152602(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-methylpheny...)
Affinity DataIC50:  314nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152593(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2-fluoropheny...)
Affinity DataIC50:  321nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50356198(CHEMBL1910222)
Affinity DataIC50:  330nMAssay Description:Inhibition of jack bean urease assessed as ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM178018((Z)-N-(3-(4-aminosulfonylphenyl)-4-methylthiazol-2...)
Affinity DataIC50:  350nMpH: 8.2Assay Description:The urease inhibitory activity of synthesized sulfonamides (3a-j) was determined by measuring the amount of ammonia produced by the indophenols metho...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM110171(Ethyl 4-[3-(2-bromobenzoyl)thioureido]benzoate (1h...)
Affinity DataIC50:  350nMpH: 8.2 T: 2°CAssay Description:The assay mixture contained 40 µL of buffer (0.01 M LiCl2, 1 mM EDTA, 0.01M K2HPO4, pH 8.2) containing 100 mM urea, 10 µL of enzyme (5U/mL)...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50521797(CHEMBL4438182)
Affinity DataIC50:  358nMAssay Description:Inhibition of jack bean urease incubated for 30 mins by indophenol methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50123235(CHEMBL3622686)
Affinity DataIC50:  370nMAssay Description:Inhibition of jack beans urease assessed as hydrolysis of urea into ammonia preincubated for 10 mins followed by urea addition measured after 10 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50253259(CHEMBL4074987)
Affinity DataIC50:  380nMAssay Description:Inhibition of jack bean urease using urea as substrate pretreated for 15 mins followed by substrate addition by phenol red based spectrophotometric m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease [D459Y,K653P](Canavalia ensiformis (Jack bean))
University Of Karachi

LigandPNGBDBM152594(2-(1-(Benzofuran-2-yl)ethylidene)-N-(2,4-difluorop...)
Affinity DataIC50:  387nMpH: 8.2Assay Description:The mixture of this enzyme inhibition assay was composed of 10 無 of enzyme (5 U/mL) and 10 無 of each test compound in the series (3a-3s) in 40 無 b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50129797(CHEMBL3629072)
Affinity DataIC50:  400nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as ammonia production incubated for 15 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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