TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 0.0130nMAssay Description:Agonist activity by measuring the [3H]thymidine uptake against Dopamine receptor D2L from ratMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 0.400nMAssay Description:In vitro effective concentration tested on HEK293 cells co-transfected with rat Dopamine receptor D2 using FLIPR assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at rat D2 receptor in HEK293 cells coexpressing Galphaqo5 by FLIPRMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:In vitro effective concentration tested on HEK293 cells co-transfected with rat Dopamine receptor D2 using FLIPR assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Agonist activity at rat D2 receptor in HEK293 cells coexpressing Galphaqo5 by FLIPRMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 1.80nMAssay Description:In vitro effective concentration tested on HEK293 cells co-transfected with ferret Dopamine receptor D2 using FLIPR assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at Rattus norvegicus (rat) dopamine D2 receptor transfected in african green monkey COS7 cells assessed as inhibition of forskolin-s...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 2.20nMAssay Description:Agonist activity by measuring the [3H]thymidine uptake against Dopamine receptor D2L from ratMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 5nMAssay Description:Activity at rat dopamine D2L receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 5.70nMAssay Description:Agonist activity by measuring the [3H]thymidine uptake against Dopamine receptor D2L from ratMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 5.70nMAssay Description:Effective concentration was determined as thymidine uptake in CHO-L6 cells transfected with the rat Dopamine receptor D2L by mitogenesis assay (intri...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 7.90nMAssay Description:Agonist activity at Rattus norvegicus (rat) dopamine D2 receptor transfected in african green monkey COS7 cells assessed as inhibition of forskolin-s...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 8nMAssay Description:In vitro effective concentration tested on HEK293 cells co-transfected with ferret Dopamine receptor D2 using FLIPR assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 8.5nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 8.70nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:Activity at rat dopamine D2L receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 9.20nMAssay Description:Effective concentration required for agonistic activity against rat D2 long receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 9.20nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2L mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 10.8nMAssay Description:In vitro effective concentration tested on HEK293 cells co-transfected with rat Dopamine receptor D2 using FLIPR assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 11nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2L mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Binding affinity of compound measured using [3H]-spiperone for the cloned human dopamine receptor D2 long (high/low affinity is given as 230/53000)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 12nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2S mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 16nMAssay Description:Effective concentration required for agonistic activity against rat Dopamine receptor D2LMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 17nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2S mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Effective concentration was determined as thymidine uptake in CHO-L6 cells transfected with the rat Dopamine receptor D2L by mitogenesis assay (intri...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Effective concentration required for agonistic activity against rat D2 long receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 19nMAssay Description:Effective concentration required for agonistic activity against rat D2 long receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 22nMAssay Description:Agonist activity at Rattus norvegicus (rat) dopamine D2 receptor transfected in african green monkey COS7 cells assessed as inhibition of forskolin-s...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 23nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 24nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 30nMAssay Description:Agonist activity at rat D2 dopamine receptor expressed in CHOK1 cells assessed as [35S]GTPgammaS binding after 90 mins by liquid scintillation counte...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 35nMAssay Description:In vitro effective concentration tested on HEK293 cells co-transfected with ferret Dopamine receptor D2 using FLIPR assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 40nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 42nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2L mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 43nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 47nMAssay Description:Binding affinity of compound measured using [3H]-spiperone for the cloned human dopamine receptor D4.4 (high/low affinity is given as 16/1300)More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 48nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2L mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at Rattus norvegicus (rat) dopamine D2 receptor transfected in african green monkey COS7 cells assessed as inhibition of forskolin-s...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 51nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 53nMAssay Description:Agonist activity at rat dopamine D2short receptor expressed in CHO-K1 cells assessed as stimulation of [35S]GTPgammaS binding by liquid scintillation...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:Agonist activity at rat dopamine D2(short) receptor expressed in CHOK1 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 55nMAssay Description:In vitro effective concentration tested on HEK293 cells co-transfected with rat Dopamine receptor D2 using FLIPR assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 58nMAssay Description:Agonist activity at rat dopamine D2(short) receptor expressed in CHOK1 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 70nMAssay Description:Activity at rat dopamine D2L receptor expressed in HEK293 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Agonist activity at rat dopamine D2(short) receptor expressed in CHOK1 cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 76nMAssay Description:Agonist activity at Rattus norvegicus (rat) dopamine D2 receptor transfected in african green monkey COS7 cells assessed as inhibition of forskolin-s...More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 79nMAssay Description:Effective concentration to stimulate rat Dopamine receptor D2S mediated [3H]-thymidine incorporation into growing cells using mitogenesis assayMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
University Centre For Pharmacy
Curated by ChEMBL
University Centre For Pharmacy
Curated by ChEMBL
Affinity DataEC50: 122nMAssay Description:Agonist activity by measuring the [3H]thymidine uptake against Dopamine receptor D2L from ratMore data for this Ligand-Target Pair