Compile Data Set for Download or QSAR
(2D       Computed 3D by Vconf -m prep )

Data curated solely by BindingDB

Found 10 hits of affinity data for UniProtKB/TrEMBL: P17252

Target (Institution)	Ligand	Target Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	pH	Temp °C
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 12	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	0.9	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	AEB071 (Sotrastaurin)	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS MMDB PC cid PC sid PDB	MMDB PDB PubMed	n/a	n/a	2.1	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 10	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	2.2	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	BIM-1 (2-[1-(3-dimethylaminopropyl)-indol-3-yl]-3-(indol-...)	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	B.MOAD CHEBI CSLS KEGG MMDB PC cid PC sid PDB	PubMed	n/a	n/a	2.3	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 11	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	7.1	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 9	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	15.0	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 5	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	73.0	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 3	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	98.0	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 4	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	>315.0	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)
Protein Kinase C, alpha Homo sapiens (Human)	maleimide derivative, 13	DrugBank GoogleScholar KEGG MMDB PDB UniProtKB/SwissProt UniProtKB/TrEMBL	CSLS PC cid PC sid	PubMed	n/a	n/a	1502.0	n/a	n/a	7.4	23
Novartis					J Med Chem. 52: 6193-6 (2009)

• Reorder this table by ec50
• Reorder this table by ic50
• Reorder this table by kd
• Reorder this table by pH
• Reorder this table by T
• Change energy unit to:  kcal/mole