Compile Data Set for Download or QSAR
maximum 50k data
Found 48 of ic50 for UniProtKB: P09958
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601761(CHEMBL5203869 | US11773078, Example 263)
Affinity DataIC50:  0.158nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601763(CHEMBL5197625 | US11773078, Example 62)
Affinity DataIC50:  0.158nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601747(CHEMBL5175553 | US11773078, Example 11)
Affinity DataIC50:  0.251nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601762(CHEMBL5190891 | US11773078, Example 369)
Affinity DataIC50:  0.501nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601704(CHEMBL5184039)
Affinity DataIC50:  0.560nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601703(CHEMBL5202322)
Affinity DataIC50:  0.560nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601759(CHEMBL5175809 | US11773078, Example 298)
Affinity DataIC50:  0.631nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601749(CHEMBL5171461 | US11773078, Example 180)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601754(CHEMBL5208861 | US11773078, Example 207)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601750(CHEMBL5182363 | US11773078, Example 41)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601757(CHEMBL5206910 | US11773078, Example 131)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601755(CHEMBL5195577 | US11773078, Example 126)
Affinity DataIC50:  1nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601760(CHEMBL5180159 | US11773078, Example 306)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601756(CHEMBL5196204 | US11773078, Example 334)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601752(CHEMBL5172689 | US11773078, Example 340)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601751(CHEMBL5200817 | US11773078, Example 339)
Affinity DataIC50:  2nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601746(CHEMBL5172764 | US11773078, Example 10)
Affinity DataIC50:  2nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601758(CHEMBL5170962 | US11773078, Example 242)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601753(CHEMBL5207406 | US11773078, Example 206)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601702(CHEMBL5199257)
Affinity DataIC50:  3nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM207839(US9266828, B)
Affinity DataIC50:  3.70nMpH: 7.5 T: 2°CAssay Description:Furin activity was measured in triplicate in wells of a 96-well plate in 0.2 ml 50 mM HEPES, pH 7.5, containing 1 mM CaCl2, 0.005% Brij-35 and 20% gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601748(CHEMBL5169887 | US11773078, Example 12)
Affinity DataIC50:  5nMAssay Description:Inhibition of Tev-FLAG-His-tagged furin (108 to 574 residues) (unknown origin) using FAM-QRVRRAVGIDK-TAMRA as substrate and measured after 2 hrsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM207838(US9266828, A)
Affinity DataIC50:  7nMpH: 7.5 T: 2°CAssay Description:Furin activity was measured in triplicate in wells of a 96-well plate in 0.2 ml 50 mM HEPES, pH 7.5, containing 1 mM CaCl2, 0.005% Brij-35 and 20% gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM207840(US9266828, C)
Affinity DataIC50:  9nMpH: 7.5 T: 2°CAssay Description:Furin activity was measured in triplicate in wells of a 96-well plate in 0.2 ml 50 mM HEPES, pH 7.5, containing 1 mM CaCl2, 0.005% Brij-35 and 20% gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50601701(CHEMBL5177253)
Affinity DataIC50:  9.5nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50399746(CHEMBL2179435)
Affinity DataIC50:  20nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50571192(CHEMBL4869416)
Affinity DataIC50:  290nMAssay Description:Inhibition of recombinant human furin ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50571193(CHEMBL4877358)
Affinity DataIC50:  290nMAssay Description:Inhibition of recombinant human furin ProteaseMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM207842(US9266828, E)
Affinity DataIC50:  300nMpH: 7.5 T: 2°CAssay Description:Furin activity was measured in triplicate in wells of a 96-well plate in 0.2 ml 50 mM HEPES, pH 7.5, containing 1 mM CaCl2, 0.005% Brij-35 and 20% gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM207841(US9266828, D)
Affinity DataIC50:  1.20E+3nMpH: 7.5 T: 2°CAssay Description:Furin activity was measured in triplicate in wells of a 96-well plate in 0.2 ml 50 mM HEPES, pH 7.5, containing 1 mM CaCl2, 0.005% Brij-35 and 20% gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM29692((2Z)-3-ethyl-2-[(E)-3-(3-ethyl-4,5-dihydro-1,3-thi...)
Affinity DataIC50:  3.15E+4nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM29692((2Z)-3-ethyl-2-[(E)-3-(3-ethyl-4,5-dihydro-1,3-thi...)
Affinity DataIC50:  3.15E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM29692((2Z)-3-ethyl-2-[(E)-3-(3-ethyl-4,5-dihydro-1,3-thi...)
Affinity DataIC50:  3.38E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM29692((2Z)-3-ethyl-2-[(E)-3-(3-ethyl-4,5-dihydro-1,3-thi...)
Affinity DataIC50:  3.38E+4nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM67896((5E)-5-(3-methylbenzylidene)-2-[N'-(1,7,7-trimethy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM71871(5,5-dimethyl-2-[(3-pyridinylamino)methylidene]cycl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM60407((5Z)-5-[[4-(dimethylamino)anilino]methylene]-1-(o-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM75777(2-[[(4-ketoquinazolin-3-yl)amino]methylene]-5,5-di...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM75778((4-Dimethylamino-phenyl)-[(4-dimethylamino-phenyl)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM74846((5Z)-1-(3-methylphenyl)-5-[(E)-3-phenylazanylprop-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM75780(5,5-Dimethyl-2-[(6-methyl-pyridin-2-ylamino)-methy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM66635(MLS000737122 | SMR000528383 | [4-[(2Z)-2-(4-amino-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Official Symbol FURIN and Name: furin (paired basic amino acid cleaving enzyme) [Homo sapiens] Other Aliases: FUR, PACE, PCSK3, SPC1 Other Designati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PCBioAssay
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50257103(5-methoxy-2-(5-nitrothiazol-2-ylthio)benzo[d]thiaz...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50257184(2-(5-nitrothiazol-2-ylthio)benzo[d]thiazole | BI-8...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of furin (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50310142(5-(5-Nitrothiazol-2-ylthio)-N-propyl-1,3,4-thiadia...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FURINMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50310148(BI-90H9 | CHEMBL611079 | N-(2-Methoxyethyl)-5-(5-n...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FURINMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50310146(BI-90H10 | CHEMBL599111 | N-(3,4-Dimethoxyphenethy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FURINMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
University Of Michigan

Curated by ChEMBL
LigandPNGBDBM50310147(BI-98A10 | CHEMBL599518 | N-sec-Butyl-5-(5-nitroth...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of FURINMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed