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Found 3 of ic50 for UniProtKB: P00514
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM50011236(CHEMBL344314 | Isoquinoline-5-sulfonic acid (2-ami...)
Affinity DataIC50:  3.60E+3nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
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TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM92674(Isoquinolinesulfonamide, CKI-7)
Affinity DataIC50:  5.50E+5nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetcAMP-dependent protein kinase type I-alpha regulatory subunit(Bos taurus)
Nagoya University School Of Medicine

LigandPNGBDBM92673(Isoquinolinesulfonamide, CKI-6)
Affinity DataIC50: >1.00E+6nMpH: 7.4 T: 2°CAssay Description:Casein kinase activities were determined under the conditions as described by Huang et al (1982).More data for this Ligand-Target Pair
In DepthDetails PubMed