Affinity DataEC50: 1.60nMAssay Description:Antagonist activity at rat recombinant 5HT3 receptor assessed as inhibition of RAMH-induced [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
Affinity DataEC50: 1.20E+4nMAssay Description:Response at rat 5-hydroxytryptamine 3a receptor expressed in xenopus oocytesMore data for this Ligand-Target Pair
Affinity DataEC50: 2.90E+4nMAssay Description:Agonist activity at rat 5HT3A expressed in Xenopus oocytes at -60 mV holding potential by electrophysiology methodMore data for this Ligand-Target Pair