Affinity DataIC50: 0.0200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0300nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0400nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0600nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0800nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0900nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Binding affinity for rat brain Angiotensin II receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.110nMAssay Description:In vivo inhibitory concentration against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.130nMAssay Description:In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.140nMAssay Description:In vivo inhibitory concentration of the compound against AT2 receptor of rat adrenal membraneMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor A/Type-1 angiotensin II receptor B/Type-2 angiotensin II receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 0.150nMAssay Description:Inhibition of [125I]AII binding to Angiotensin II receptor, type 1 of rat mesenteric arteriesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.150nMAssay Description:In vitro displacement of [125I]angiotensin II from rat liver (Angiotensin 1 receptor) membrane preparationMore data for this Ligand-Target Pair
Affinity DataIC50: 0.160nMAssay Description:Tested for inhibition of [125I]- AII specific binding to rat mesenteric arteries, expressed as IC50More data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:In vivo inhibitory concentration of the compound against Angiotensin II, type 2 of rat midbrain membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Compound was evaluated for the in vitro inhibition of specific binding of [125I]-A II to Angiotensin II receptor, type 1 from rat adrenal membranes.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:In vitro binding affinity at Angiotensin II Type 1 receptor in rat liver membrane by [125I]AII displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Specific binding inhibition of [125I]AII to Angiotensin II receptor, type 1 in rat liver membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Concentration required for 50% inhibition of [125I]- AII binding to rat liver membrane preparation (AT1)More data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity against Angiotensin II receptor, type 1 using [125I]Sar-Ile8-AII in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Binding affinity against Angiotensin II receptor, type 1 using [125I]Sar-Ile8-AII in rat liver membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory activity against rat Angiotensin II receptor, type 1 expressed in CHO cellsMore data for this Ligand-Target Pair