Compile Data Set for Download or QSAR
maximum 50k data
Found 28 of ec50 data for polymerid = 49000349
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM82235(Gastrin I | Gastrin-17 | Gastrin-I-(1-17))
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50348753(CHEMBL1806528)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50348752(CHEMBL1807150)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092405((S)-N-((S)-1-Carbamoyl-2-phenyl-ethyl)-3-((S)-2-{[...)
Affinity DataEC50:  0.400nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50348756(CHEMBL1806532)
Affinity DataEC50:  0.410nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50024321(3-{2-[2-(3-tert-Butoxycarbonylamino-propionylamino...)
Affinity DataEC50:  0.430nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092408(CHEMBL120150 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2...)
Affinity DataEC50:  0.560nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.630nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM21147((3S)-3-[(2S)-2-[(2S)-2-{2-[(2S)-2-[(2S)-2-[(3S)-3-...)
Affinity DataEC50:  0.630nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50002477((S)-3-{(S)-2-[(S)-2-tert-Butoxycarbonylamino-3-(1H...)
Affinity DataEC50:  1nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50549228(CHEMBL4758706)
Affinity DataEC50:  1.30nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50024317(3-{2-[2-Amino-3-(1H-indol-3-yl)-propionylamino]-4-...)
Affinity DataEC50:  1.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092384(CHEMBL100538 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2...)
Affinity DataEC50:  1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092398((S)-3-((S)-2-{[(S)-2-tert-Butoxycarbonylamino-3-(1...)
Affinity DataEC50:  1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50056453(3-(2-{[2-tert-Butoxycarbonylamino-3-(1H-indol-3-yl...)
Affinity DataEC50:  1.5nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092391(3-(2-{[2-(2-Carbamoyl-acetylamino)-3-(1H-indol-3-y...)
Affinity DataEC50:  1.64nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50549226(CHEMBL4795913)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50549227(CHEMBL4759105)
Affinity DataEC50:  1.90nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092389(CHEMBL321456 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-(2...)
Affinity DataEC50:  2nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092399(3-(2-{[2-(2-Benzylcarbamoyl-acetylamino)-3-(1H-ind...)
Affinity DataEC50:  3.30nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092393(3-(2-{[2-(2-{2-[2-tert-Butoxycarbonylamino-3-(4-su...)
Affinity DataEC50:  3.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50056448(CHEMBL2371221 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataEC50:  4nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50056455(CHEMBL348344 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[...)
Affinity DataEC50:  7nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50056449(CHEMBL2371222 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{...)
Affinity DataEC50:  7nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092401(CHEMBL177799 | N-(1-Carbamoyl-2-phenyl-ethyl)-3-{[...)
Affinity DataEC50:  7nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50092395(3-{2-[2-{[9-tert-Butoxycarbonylamino-3-butyl-2,5,8...)
Affinity DataEC50:  17nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50026690(2-[2-(2-{2-[2-{2-[2-(2-Amino-3-phenyl-propionylami...)
Affinity DataEC50:  1.00E+3nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana

Curated by ChEMBL
LigandPNGBDBM50037873(CBS-2 | CHEMBL341130)
Affinity DataEC50:  2.00E+5nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed