TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.170nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.270nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.330nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.400nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.410nMAssay Description:Agonist activity at gastrin receptor in rat AR4-2J cells assessed as intracellular calcium mobilization by fluorescence assayMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.430nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.560nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.630nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 0.630nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.30nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.5nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.64nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.70nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.90nMAssay Description:Agonist activity at rat CCK2R expressed in rat AR42J cells assessed as intracellular calcium mobilization measured after 24 hrs by Fluo-4AM dye based...More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 2nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 3.30nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 3.40nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 4nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Effective concentration for the stimulation of Inositol Phosphate accumulation in CHO cells expressing wild-type Cholecystokinin type B receptorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 7nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 17nMAssay Description:Affinity against Cholecystokinin type B receptor expressed in CHO cells on rat brain.More data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 1.00E+3nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(RAT)
University Medical Centre Ljubljana
Curated by ChEMBL
University Medical Centre Ljubljana
Curated by ChEMBL
Affinity DataEC50: 2.00E+5nMAssay Description:Tested for the 50% inhibition level against [125I]- gastrin binding in AR42J cellsMore data for this Ligand-Target Pair