Compile Data Set for Download or QSAR
maximum 50k data
Found 37 of ic50 for UniProtKB: P08485
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50176065(4-DAMP | 4-Diphenylacetoxy-1,1-dimethyl-piperidini...)
Affinity DataIC50:  1.90nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50064609(6-acetoxy-8-azonia-bicyclo[3.2.1]octane | Acetic a...)
Affinity DataIC50:  11nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50577262(CHEMBL4853244)
Affinity DataIC50:  57nMAssay Description:Displacement of [3H]NMS from rat muscarinic receptor M4 expressed in CHO cell membranes incubated for 3 hrs by radiometric scintillation counting ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50596229(CHEMBL5205163)
Affinity DataIC50:  81nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50596229(CHEMBL5205163)
Affinity DataIC50:  81nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50577263(CHEMBL4850236)
Affinity DataIC50:  145nMAssay Description:Displacement of [3H]NMS from rat muscarinic receptor M4 expressed in CHO cell membranes incubated for 3 hrs by radiometric scintillation counting ana...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50596242(CHEMBL5185664)
Affinity DataIC50:  228nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50004656((2-Carbamoyloxy-ethyl)-trimethyl-ammonium | (2-Car...)
Affinity DataIC50:  230nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50006243(((2S,4R,5S)-4-Hydroxy-5-methyl-tetrahydro-furan-2-...)
Affinity DataIC50:  470nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50240543(CHEMBL4096589)
Affinity DataIC50:  478nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50263887(1-(1'-(2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-b...)
Affinity DataIC50:  493nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50596230(CHEMBL5178468)
Affinity DataIC50:  525nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50596230(CHEMBL5178468)
Affinity DataIC50:  530nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50240543(CHEMBL4096589)
Affinity DataIC50:  560nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50240546(CHEMBL4085711)
Affinity DataIC50:  562nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50240546(CHEMBL4085711)
Affinity DataIC50:  590nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50577261(CHEMBL4849905)
Affinity DataIC50:  597nMAssay Description:Displacement of [3H]NMS from rat muscarinic receptor M4 expressed in CHO cell membranes incubated for 3 hrs by radiometric scintillation counting ana...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM48918(2-acetoxypropyl(trimethyl)ammonium;chloride | 2-ac...)
Affinity DataIC50:  700nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50268343(CHEMBL4096727)
Affinity DataIC50:  1.00E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373835(CHEMBL256202)
Affinity DataIC50:  5.10E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50424114(CHEMBL2315675)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50424114(CHEMBL2315675)
Affinity DataIC50:  5.20E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373841(CHEMBL270580)
Affinity DataIC50:  7.90E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50424117(CHEMBL2315680)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50424122(CHEMBL2315676)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373834(CHEMBL255169)
Affinity DataIC50:  1.80E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373836(CHEMBL271704)
Affinity DataIC50:  2.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50445223(CHEMBL3105208)
Affinity DataIC50: >3.00E+4nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50445222(CHEMBL3105228)
Affinity DataIC50: >3.00E+4nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50231856(CHEMBL271519 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50:  6.60E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373833(CHEMBL404874)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373832(CHEMBL429780)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373840(CHEMBL258281)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373838(CHEMBL258335)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373839(CHEMBL438706)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50373837(CHEMBL429320)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo

Curated by ChEMBL
LigandPNGBDBM50231845(CHEMBL255523 | N-(3-chloro-4-(4-ethylpiperazin-1-y...)
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed