TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 57nMAssay Description:Displacement of [3H]NMS from rat muscarinic receptor M4 expressed in CHO cell membranes incubated for 3 hrs by radiometric scintillation counting ana...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 81nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 145nMAssay Description:Displacement of [3H]NMS from rat muscarinic receptor M4 expressed in CHO cell membranes incubated for 3 hrs by radiometric scintillation counting ana...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 228nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 470nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 478nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 493nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 525nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 530nMAssay Description:Inhibition of rat muscarinic acetylcholine M4 receptor expressed in CHO cells co-expressing Gqi5 in the presence of acetylcholine at EC80 concentrati...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 560nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 562nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Antagonist activity at rat M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 597nMAssay Description:Displacement of [3H]NMS from rat muscarinic receptor M4 expressed in CHO cell membranes incubated for 3 hrs by radiometric scintillation counting ana...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 700nMAssay Description:Inhibitory activity against [3H]-cyclic AMP accumulation in CHO transfected cells mediated by Muscarinic acetylcholine receptor M4More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 5.10E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 7.90E+3nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells assessed as inhibition of Ach-induced calcium responseMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 1.80E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Negative allosteric modulation of rat muscarinic acetylcholine receptor M4 expressed in CHO cells assessed as inhibition of acetylcholine-induced cal...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: 6.60E+4nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M4(RAT)
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Universit£ degli Studi di Urbino Carlo Bo
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M4 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair